In order to address the urgent need to develop well-qualified research scientists in a multidisciplinary field between chemistry and biology, Chemical Biology Program has been established at the Chulabhorn Graduate Institute. Some of our current Ph.D. staffs have participated in the Chemical Biology Program as core curriculum members and have actively produced highly motivated graduates at both the Master’s and doctor of philosophy levels to lead research teams to tackle the research problems at the interface between chemistry and biology, especially in drug discovery and development.