Publications (2008 – present)

2018

Akkachairin B, Tummatorn J, Khamsuwan N, Thongsornkleeb C, Ruchirawat S. Domino N₂–Extrusion–Cyclization of Alkynylarylketone Derivatives for the Synthesis of Indoloquinolines and Carbocycle-fused Quinolines. J. Org. Chem. 2018; 83: 11254-11268. Abstract

Nimnual P, Norseeda K, Akkachairin B, Tummatorn J, Laohapaisan P, Supantanapong N, Chuangsoongnern P, Thongsornkleeb C, Sittihan S, Ruchirawat S, Rodphon W. Synthesis of β‐Naphthols and Naphthofuranones from ortho‐Alkynylarylketones viaSequential AgTFA‐catalyzed Ketonization–Intramolecular Aldol Condensation: A Total Synthesis of Negundin A. Asian J. Org. Chem. 2018; 7: 932-945. Abstract

Disadee W, Ruchirawat S. One-pot Cascade Synthesis of Azabicycles via the Nitro-Mannich Reaction and N-Alkylation. Org. Biomol. Chem. 2018; 16: 707-711. Abstract

Pongpamorn P, Wan-erlor S, Ruchirawat S, Thasana N. Semi-synthetic Studies of α-Onocerin Derivative for Cytotoxicity. Phytochem. Lett. 2018; 23: 106-115.Abstract

2017

Chuangsoongnern P, Surinrach C, Tummatorn J, Thongsornkleeb C, Ruchirawat S. Iodine-mediated Cyclization of ortho-Alkynylaryl Ketones for the Synthesis of Indenone Derivatives. Eur. J. Org. Chem. 2017; 2017: 5102-5109. Abstract

Ieawsuwan W, Ruchirawat S. PIFA–BF₃•OEt₂ Mediated Intramolecular Regioselective Domino Cyclization of Ynamides: A Novel Method for the Synthesis of Tetrahydroisoquinoline-oxazol-2(3H)-ones. Bioorg. Med. Chem. 2017; 25: 2856-2867.Abstract

Ruchirawat S, Disadee W. A One-pot, Metal-free Approach to Bicyclic 2-Pyridones. Org. Chem. Front. 2017; 4: 2026-2030. Abstract

Akkachairin B, Tummatorn J, Supantanapong N, Nimnual P, Thongsornkleeb C, Ruchirawat S. Silver-catalyzed Cyclization of ortho-Carbonylarylacetylenols for the Synthesis of Dihydronaphthofurans. J. Org. Chem. 2017; 82: 3727-3740. Abstract

Tangdenpaisal K, Chuayboonsong K, Ruchirawat S, Ploypradith P. A Divergent Strategy for the Diastereoselective Synthesis of the Tricyclic 6,7-Diaryl-tetrahydro-6H-benzo[c]chromene Core via Pt(IV)-catalyzed Cycloaddition of ortho-Quinone Methides and Olefin Ring-closing Metathesis. J. Org. Chem. 2017; 82: 2672-2688. Abstract

Nealmongkol P, Calmes J, Ruchirawat S, Thasana N. Synthesis of Phenanthridinones using Cu- or Pd-mediated C–N bond formation. Tetrahedron 2017; 73: 735-741. Abstract

2016

Pongpamorn P, Wan-erlor S, Ruchirawat S, Thasana N. Lycoclavatumide and 8β,11α-Dihydroxylycopodine, a New Fawcettimine and Lycopodine-type Alkaloid from Lycopodium clavatum. Tetrahedron 2016; 72: 7065-7069. Abstract

Yasamut K, Jongcharoenkamol J, Ruchirawat S, Ploypradith P. A Modified Cu(0)-Cu(I)-mediated C_aryl-C_aryl Ullmann Coupling for the Synthesis of Biaryls. Tetrahedron 2016; 72: 5994-6000. Abstract

Nilsu T, Thorroad S, Ruchirawat S, Thasana N. New Lycopodium Alkaloids from Thai and Philippine Huperzia squarrosa. Planta Med. 2016; 82: 1046-1050. Abstract

Norseeda K, Tummatorn J, Krajangsri S, Thongsornkleeb C, Ruchirawat S. Synthesis of 6-Alkyl-6 H-benzo[c]chromene Derivatives by Cyclization/Selective Ether Cleavage in One Pot: Total Synthesis of Cannabinol. Asian J. Org. Chem. 2016; 5: 792-800. Abstract

2015

Theppawong A, Ploypradith P, Chuawong P, Ruchirawat S, Chittchang M. Facile and Divergent Synthesis of Lamellarins and Lactam-containing Derivatives with Improved Drug Likeness and Biological Activities. Chem Asian J. 2015; 2631-2650. Abstract

Nimnual P, Tummatorn J, Thongsornkleeb C, Ruchirawat S. Utility of Nitrogen Extrusion of Azido Complexes for the Synthesis of Nitriles, Benzoxazoles, and Benzisoxazoles. J. Org. Chem. 2015; 80: 8657-8667. Abstract

Tummatorn J, Poonsilp P, Nimnual P, Janprasit J, Thongsornkleeb C, Ruchirawat S. Regioselective Synthesis of 3-Bromoquinoline Derivatives and Diastereoselective Synthesis of Tetrahydroquinolines via Acid-Promoted Rearrangement of Arylmethyl Azides. J. Org. Chem. 2015; 80: 4516-4525. Abstract

Aroonkit P, Thongsornkleeb C, Tummatorn J, Krajangsri S, Mungthin M, Ruchirawat S. Synthesis of Isocryptolepine Analogues and Their Structure-activity Relationship Studies as Antiplasmodial and Antiproliferative Agents. Eur. J. Med. Chem. 2015; 94: 56-62. Abstract

Tangdenpaisal K, Worayuthakarn R, Karnkla S, Ploypradith P, Intachote P, Sengsai S, Saimanee B, Ruchirawat S, Chittchang M. Designing New Analogs for Streamlining the Structure of Cytotoxic Lamellarin Natural Products. Chem. Asian J. 2015; 10: 925-937. Abstract

Tangdenpaisal K, Chuayboonsong K, Sukjarean P, Katesampao V, Noiphrom N, Ruchirawat S, Ploypradith P. Synthesis of C4–C5 Cycloalkyl-fused and C6-modified Chromans via ortho-Quinone Methides. Chem. Asian J. 2015; 10: 1050-1064. Abstract

Tummatorn J, Thongsornkleeb C, Ruchirawat S, Thongarama P, Kaewmeea B. Convenient and Direct Azidation of sec-Benzyl Alcohols by Trimethylsilyl Azide with Bismuth(III) Triflate Catalyst. Synthesis 2015; 47: 325-329. Abstract

2014

Thorroad S, Worawittayanont P, Khunnawutmanotham N, Chimnoi N, Jumruksa A, Ruchirawat S, Thasana N. Three New Lycopoium Alkaloids from Huperzia carinata and H. squarrosa. Tetrahedron 2014; 70: 8017-8022. Abstract

Tangdenpaisal K, Ruchirawat S, Ploypradith P. Synthesis of the Thyroid Hormone Analog GC-1 via Bi(OTf)₃-catalyzed Benzylation. Tetrahedron 2014; 70: 6789-6795. Abstract

Tummatorn J, Krajangsri S, Norseeda K, Thongsornkleeb C, Ruchirawat S. A New Synthetic Approach to 6-Unsubstituted Phenanthridine and Phenanthridine-like Compounds under Mild and Metal-free Conditions. Org. Biomol. Chem. 2014; 12: 5077-5081. Abstract

Tummatorn J, Gleeson MP, Krajangsri S, Thongsornkleeb C, Ruchirawat S. ZrCl₄-promoted Facile Synthesis of Indole Derivatives. RSC Adv. 2014; 4: 20048-20052. Abstract

Worayuthakarn R, Boonya-udtayan S, Ruchirawat S, Thasana N. Total Synthesis of Unsymmetrical Benzils, Scandione and Calophione A. Eur. J. Org. Chem. 2014; 2496-2507. Abstract

2013

Nealmongkol P, Tangdenpaisal K, Ruchirawat S, Thasana N. Cu(I)-mediated Lactone Formation in Subcritical Water: A Benign Synthesis of Benzopyranones and Urolithins A-C. Tetrahedron 2013; 69: 9277-9283. Abstract

Sarnpitak P, Trongchit K, Kostenko Y, Sathalalai S, Gleeson MP, Ruchirawat S, Ploypradith P. Synthesis of Substituted 2-Arylindanes from E-(2-Stilbenyl)methanols via Lewis Acid-mediated Cyclization and Nucleophililc Transfer from Trialkylsilyl Reagents. J. Org. Chem. 2013; 78: 8281-8296. Abstract

Tummatorn J, Thongsornkleeb C, Ruchirawat S, Gettongsong T. Synthesis of 2,4-Unsubstituted Quinoline-3-carboxylic Acid Ethyl Esters from Arylmethyl Azides via a Domino Process. Org. Biomol. Chem. 2013; 11: 1463-1467. Abstract

Tangdenpaisal K, Phakhodee W, Ruchirawat S, Ploypradith P. Facile Synthesis of Diarylmethanes via Quinone Methides. Tetrahedron 2013; 69: 933-941. Abstract

2012

Boonya-Udtayan S, Eno M, Ruchirawat S, Mahidol C, Thasana N. Palladium-catalyzed Intramolecular C–H Amidation: Synthesis and Biological Activities of Indolobenzazocin-8-ones. Tetrahedron 2012; 68: 10293-10301.Abstract

Tummatorn J, Thongsornkleeb C, Ruchirawat S. Acid-promoted Rearrangement of Arylmethyl Azides: Applications toward the Synthesis of N-Arylmethyl Arenes and Polycyclic Heteroaromatic Compounds. Tetrahedron 2012; 68: 4732-4739. Abstract

Worayuthakarn R, Nealmongkol P, Ruchirawat S, Thasana N. Synthesis of Benzoindoloquinolizines via a Cu(I)-mediated C– N Bond Formation. Tetrahedron 2012; 68: 2864-2875. Abstract

Wittayalai S, Sathalalai S, Thorroad S, Worawittayanon P, Ruchirawat S, Thasana N. Lycophlegmariols A-D: Cytotoxic Serratene Triterpenoids from the Club Moss Lycopodium phlegmaria L. Phytochemistry 2012; 76: 117-123. Abstract

2011

Disadee W, Ploypradith P, Aree T, Chaichit N, Ruchirawat S. A Novel Approach for the Synthesis of Lophocladines A, B and C1 Analogues. Tetrahedron Lett. 2011; 52: 6142-6144. Abstract

Radomkit S, Sarnpitak P, Tummatorn J, Batsomboon P, Ruchirawat S, Ploypradith P. Pt(IV)-catalyzed Generation and [4+2]-Cycloaddition Reactions of O-Quinone Methides. Tetrahedron 2011; 67: 3904-3914. Abstract

Gleeson MP, Deechongkit S, Ruchirawat S. Molecular Dynamics Investigation of Psalmopeotoxin I. Probing the Relationship between 3D Structure, Anti-malarial Activity and Thermal Stability. J. Mol. Model. 2011; 17: 769-775. Abstract

2010

Boonya-Udtayan S, Yotapan N, Woo C, Bruns CJ, Ruchirawat S, Thasana N. Synthesis and Biological Activities of Azalamellarins. Chem. Asian J. 2010; 5: 2113-2123. Abstract

Chittchang M, Gleeson MP, Ploypradith P, Ruchirawat S. Assessing the Drug-likeness of Lamellarins, a Marine-derived Natural Product Class with Diverse Oncological Activities. Eur. J. Med. Chem. 2010; 45: 2165-2172. Abstract

Kamolkijkarn P, Prasertdee T, Netirojjanakul C, Sarnpitak P, Ruchirawat S, Deechongkit S. Synthesis, Biophysical, and Biological Studies of Wild-type and Mutant Psalmopeotoxins – Anti-malarial Cysteine Knot Peptides from Psalmopoeus cambridgei. Peptides 2010; 31: 533-540. Abstract

Tummatorn J, Ruchirawat S, Ploypradith P. A Convergent General Strategy for the Functionalized 2-Aryl Cycloalkylfused Chromans: Intramolecular Hetero-Diels-Alder Reactions of ortho-Quinone Methides. Chem. Eur. J. 2010; 16: 1445-1448. Abstract

2009

Tangdenpaisal K, Sualek S, Ruchirawat S, Ploypradith P. Factors Affecting Orthogonality in the Deprotection of 2,4-Di-protected Aromatic Ethers Employing Solid-supported Acids. Tetrahedron 2009; 65: 4316-4325. Abstract

Batsomboon P, Phakhodee W, Ruchirawat S, Ploypradith P. Generation of ortho-Quinone Methides by p -TsOH on Silica and Their Hetero-Diels-Alder Reactions with Styrenes. J. Org. Chem. 2009; 74: 4009-4012. Abstract

Chittchang M, Batsomboon P, Ruchirawat S, Ploypradith P. Cytotoxicities and Structure-activity Relationships of Natural and Unnatural Lamellarins toward Cancer Cell Lines. ChemMedChem 2009; 4: 457-465. Abstract

Phakhodee W, Ploypradith P, Sahakitpichan P, Ruchirawat S. A New Synthetic Approach towards Isoquinobenzazepinone and Isoindolinobenzazepinone using Acid-mediated Cyclisation and Heck Reaction. Tetrahedron 2009 ; 65: 351-356. Abstract

2008

Worayuthakarn R, Boonya-udtayan S, Arom-oon E, Ploypradith P, Ruchirawat S, Thasana N. Synthesis of Unsymmetrical Benzil Licoagrodione. J. Org. Chem. 2008; 73: 7432-7435. Abstract

Phakhodee W, Sahakitpichan P, Deechongkit S, Ruchirawat S. Investigation of the Acid-mediated Cyclisation of Amide Acetal for the Synthesis of Benzazepinone. Heterocycles 2008; 75: 1963-1970. Abstract

Thasana N, Bjerke-Kroll B, Ruchirawat S. A Facile Synthesis of Telisatin A via Microwave-promoted Annulation and Reformatsky Reaction. Synlett 2008; 505-508. Abstract